SCHEMBL9638116

SCHEMBL9638116

CCCCc1cc(C(CC)c2nc3ccc(C(=O)O)cc3[nH]2)ccc1-c1ccccc1C#N

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLKL Q8NB16 3/20 0.45
MPL P40238 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 1/20 0.38
HSP90AA1 P07900 1/20 0.37
ESR2 Q92731 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
APEX1 P27695 1/20 0.36
S1PR1 P21453 2/20 0.36
S1PR3 Q99500 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
HPGD P15428 1/20 0.35
APLNR P35414 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
TOP2A P11388 1/20 0.34
S1PR4 O95977 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9637468 0.76 PARP1 (0.39) HPGD
SCHEMBL9637462 0.75 BRS3 (0.37) APLNR
SCHEMBL9493716 0.71 BRS3 (0.39)
SCHEMBL3172738 0.70 CHEK2 (0.56) ALDH1A1HSP90AA1ESR2TDP1HPGD
SCHEMBL14089938 0.70 ALDH1A1 (0.45) ALDH1A1HPGD
SCHEMBL2932936 0.68 AKR1C3 (0.47) MPLALDH1A1MAPK1HSP90AA1ESR2
SCHEMBL3813964 0.67 MLKL (0.59) MLKLALDH1A1MAPK1HSP90AA1ESR2
SCHEMBL8906012 0.67 APEX1 (0.71) MPLALDH1A1MAPK1HSP90AA1ESR2
SCHEMBL9492881 0.66 BRS3 (0.34)
SCHEMBL17263165 0.66 MLKL (0.62) MLKLALDH1A1MAPK1HSP90AA1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5128356-A Angiotensin antagonist; cardiovascular disorders TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-07-07 US disclosed