SCHEMBL9640355

SCHEMBL9640355

CCON=C(C)C1=CC=CN(Cc2ccccc2)C1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.34
MAPK1 P28482 1/20 0.34
HTT P42858 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAPT P10636 1/20 0.33
ALDH1A1 P00352 1/20 0.33
S1PR3 Q99500 1/20 0.33
PPARG P37231 5/20 0.32
PPARA Q07869 4/20 0.32
DRD4 P21917 1/20 0.32
HPGD P15428 1/20 0.32
GAA P10253 1/20 0.32
ADRA1A P35348 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL9593810 0.99 LMNA (0.33) LMNAMAPK1HTTL3MBTL1NPC1
SCHEMBL9641212 0.87 HRH3 (0.34) MAPTALDH1A1S1PR3GAA
Bromide SCHEMBL9595283 0.86 HRH3 (0.33) MAPTALDH1A1S1PR3GAA
SCHEMBL9640334 0.83 CYP2D6 (0.35) LMNAMAPK1SMN1; SMN2MAPTALDH1A1
Bromide SCHEMBL9595609 0.82 CYP2D6 (0.35) LMNAMAPK1SMN1; SMN2MAPTALDH1A1
SCHEMBL27814642 0.77 LMNA (0.43) LMNAL3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL9641429 0.76
SCHEMBL9640312 0.75 TSHR (0.34) HTTL3MBTL1
Bromide SCHEMBL9595302 0.74 TSHR (0.33) HTTL3MBTL1
Iodide SCHEMBL9593224 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0288394-B1 1,2,5,6-TETRAHYDROPYRIDINES, PROCESS FOR THEIR PREPARATION, THEIR USE AS MEDICINES AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1992-09-09 EP disclosed
EP-0288394-A2 1,2,5,6-Tetrahydropyridines, process for their preparation, their use as medicines and compositions containing them ROUSSEL-UCLAF (FR) 1988-10-26 EP disclosed