Bromide

Bromide

SCHEMBL9595609

Br.CC(=NO)C1=CC=CN(Cc2ccccc2)C1

nearest known ligand 0.35

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 known ✓ Q99720 1/20 0.32
CYP2D6 P10635 2/20 0.35
TSHR P16473 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP2C19 P33261 1/20 0.35
GAA P10253 1/20 0.34
LMNA P02545 3/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
MC4R P32245 1/20 0.31
NOS2 P35228 1/20 0.31
ALDH1A1 P00352 1/20 0.31
BRD4 O60885 1/20 0.31
POLB P06746 1/20 0.30
MAPT P10636 1/20 0.30
MAPK1 P28482 1/20 0.30
PPARG P37231 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9640334 0.99 CYP2D6 (0.35) CYP2D6TSHRMEN1KMT2ACYP2C19
Bromide SCHEMBL9595283 0.85 HRH3 (0.33) CYP2D6TSHRMEN1KMT2AGAA
SCHEMBL9641212 0.84 HRH3 (0.34) CYP2D6TSHRMEN1KMT2AGAA
Bromide SCHEMBL9595302 0.84 TSHR (0.33) TSHRMEN1KMT2ASIGMAR1POLB
SCHEMBL9640312 0.82 TSHR (0.34) TSHRMEN1KMT2ASIGMAR1MC4R
SCHEMBL9640355 0.82 LMNA (0.34) GAALMNASMN1; SMN2ALDH1A1MAPT
SCHEMBL27814642 0.81 LMNA (0.43) CYP2D6TSHRKMT2ACYP2C19LMNA
SCHEMBL2805436 0.78 CCR2 (0.39) CYP2D6TSHRMEN1KMT2ACYP2C19
Trichloroacetic Acid SCHEMBL27834532 0.76 LMNA (0.39) CYP2D6TSHRKMT2ALMNASMN1; SMN2
SCHEMBL2353804 0.75 PARP1 (0.40) CYP2D6MEN1KMT2AGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5219873-A Treating Alzheimer*s disease, memory disorders ROUSSEL UCLAF (FR) 1993-06-15 US disclosed