SCHEMBL9640334

SCHEMBL9640334

CC(=NO)C1=CC=CN(Cc2ccccc2)C1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.35
TSHR P16473 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP2C19 P33261 1/20 0.35
GAA P10253 1/20 0.35
SIGMAR1 Q99720 1/20 0.33
LMNA P02545 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MC4R P32245 1/20 0.32
ALDH1A1 P00352 1/20 0.32
BRD4 O60885 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
PPARG P37231 1/20 0.31
PPARA Q07869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL9595609 0.99 CYP2D6 (0.35) CYP2D6TSHRMEN1KMT2ACYP2C19
SCHEMBL9641212 0.85 HRH3 (0.34) CYP2D6TSHRMEN1KMT2AGAA
Bromide SCHEMBL9595283 0.84 HRH3 (0.33) CYP2D6TSHRMEN1KMT2AGAA
SCHEMBL9640312 0.83 TSHR (0.34) TSHRMEN1KMT2ASIGMAR1MC4R
SCHEMBL9640355 0.83 LMNA (0.34) GAALMNASMN1; SMN2ALDH1A1MAPT
SCHEMBL27814642 0.82 LMNA (0.43) CYP2D6TSHRKMT2ACYP2C19LMNA
Bromide SCHEMBL9595302 0.82 TSHR (0.33) TSHRMEN1KMT2ASIGMAR1POLB
SCHEMBL2805436 0.79 CCR2 (0.39) CYP2D6TSHRMEN1KMT2ACYP2C19
Trichloroacetic Acid SCHEMBL27834532 0.77 LMNA (0.39) CYP2D6TSHRKMT2ALMNASMN1; SMN2
SCHEMBL2353804 0.77 PARP1 (0.40) CYP2D6MEN1KMT2AGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0288394-B1 1,2,5,6-TETRAHYDROPYRIDINES, PROCESS FOR THEIR PREPARATION, THEIR USE AS MEDICINES AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1992-09-09 EP disclosed
EP-0288394-A2 1,2,5,6-Tetrahydropyridines, process for their preparation, their use as medicines and compositions containing them ROUSSEL-UCLAF (FR) 1988-10-26 EP disclosed