SCHEMBL9645573

SCHEMBL9645573

CCCCCN(CCCCC)C(=O)C(CCC(=O)OC)CSc1ccc(C(C)=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCKAR P32238 1/20 0.39
CCKBR P32239 10/20 0.39
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38
LMNA P02545 2/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
HIF1A Q16665 1/20 0.37
ALDH1A1 P00352 1/20 0.37
SLCO1B3 Q9NPD5 1/20 0.37
SLCO1B1 Q9Y6L6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9645652 0.84 CCKBR (0.40) CCKARCCKBRLMNACYP3A4CYP2C9
SCHEMBL9558864 0.83 CCKBR (0.48) CCKBRLMNACYP3A4CYP2C9ALDH1A1
SCHEMBL9644811 0.83 CCKAR (0.48) CCKARCCKBRTHRBLMNACYP3A4
SCHEMBL9645565 0.80 THRA (0.44) CCKARCCKBRTHRATHRBLMNA
SCHEMBL9645604 0.77 CCKBR (0.44) CCKARCCKBRLMNACYP3A4CYP2C9
SCHEMBL9558991 0.75 PLA2G2A (0.42) CCKBRLMNACYP3A4CYP2C9
SCHEMBL9646243 0.69 MCHR1 (0.48) CCKBRTHRATHRBLMNACYP3A4
SCHEMBL9646313 0.68 CCKBR (0.41) CCKARCCKBRLMNACYP3A4CYP2C9
SCHEMBL9644737 0.67 THRA (0.46) CCKARCCKBRTHRATHRB
SCHEMBL2011642 0.66 HPGD (0.52) LMNACYP3A4CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0508004-A1 Phenylsulfonylalkanoic acid compounds Kissei Pharmaceutical Co., Ltd. (JP) 1992-10-14 EP disclosed
US-5145869-A Treatment of irritable bowel syndrome, dyskinesia, pancreatist; hormone inhibitors KISSEI PHARMACEUTICAL CO., LTD. (JP) 1992-09-08 US disclosed