SCHEMBL9646243

SCHEMBL9646243

CCCCCN(CCCCC)C(=O)C(CCC(=O)OC)CS(=O)(=O)c1ccc(C)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.48
PLA2G2C Q5R387 1/20 0.44
CCKBR P32239 1/20 0.41
THRA P10827 1/20 0.41
THRB P10828 1/20 0.41
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 5/20 0.40
CYP2C9 P11712 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
POLB P06746 1/20 0.39
MAPK1 P28482 1/20 0.39
MAPT P10636 1/20 0.37
LMNA P02545 2/20 0.37
MMP1 P03956 1/20 0.37
ALB P02768 1/20 0.36
TSHR P16473 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9645565 0.89 THRA (0.44) MCHR1PLA2G2CCCKBRTHRATHRB
SCHEMBL9646092 0.85 LMNA (0.48) CCKBRTHRBALDH1A1CYP2C9CYP3A4
SCHEMBL9558960 0.81 CCKBR (0.46) CCKBRALDH1A1MMP1
SCHEMBL9646313 0.80 CCKBR (0.41) MCHR1CCKBRALDH1A1CYP2C9CYP3A4
SCHEMBL9559158 0.79 GAA (0.48) CCKBRKMT2AALDH1A1LMNAMMP1
SCHEMBL9559024 0.79 CCKBR (0.46) CCKBRALDH1A1MMP1
SCHEMBL9646074 0.79 CCKBR (0.44) CCKBRTHRBALDH1A1CYP2C9CYP3A4
SCHEMBL9558525 0.77 ALDH1A1 (0.43) CCKBRALDH1A1LMNAMMP1
SCHEMBL9644737 0.77 THRA (0.46) CCKBRTHRATHRBMMP1
SCHEMBL9558853 0.77 ALDH1A1 (0.43) CCKBRALDH1A1LMNAMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0508004-A1 Phenylsulfonylalkanoic acid compounds Kissei Pharmaceutical Co., Ltd. (JP) 1992-10-14 EP disclosed
US-5145869-A Treatment of irritable bowel syndrome, dyskinesia, pancreatist; hormone inhibitors KISSEI PHARMACEUTICAL CO., LTD. (JP) 1992-09-08 US disclosed