SCHEMBL9645565

SCHEMBL9645565

CCCCCN(CCCCC)C(=O)C(CCC(=O)OC)CS(=O)(=O)c1ccc(C(C)=O)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.44
THRB P10828 1/20 0.44
LMNA P02545 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
HIF1A Q16665 1/20 0.39
ALDH1A1 P00352 1/20 0.39
SLCO1B3 Q9NPD5 1/20 0.39
SLCO1B1 Q9Y6L6 1/20 0.39
CCKAR P32238 1/20 0.38
CCKBR P32239 7/20 0.38
PLA2G2C Q5R387 1/20 0.37
MCHR1 Q99705 1/20 0.36
MMP1 P03956 3/20 0.36
MMP2 P08253 2/20 0.36
MMP3 P08254 2/20 0.36
MMP9 P14780 2/20 0.36
MMP8 P22894 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9646243 0.89 MCHR1 (0.48) THRATHRBLMNACYP3A4CYP2C9
SCHEMBL9644737 0.88 THRA (0.46) THRATHRBCCKARCCKBRMMP1
SCHEMBL9646092 0.84 LMNA (0.48) THRBLMNACYP3A4CYP2C9TSHR
SCHEMBL9645573 0.80 CCKAR (0.39) THRATHRBLMNACYP3A4CYP2C9
SCHEMBL9558960 0.79 CCKBR (0.46) ALDH1A1CCKARCCKBRMMP1
SCHEMBL9559024 0.77 CCKBR (0.46) ALDH1A1CCKBRMMP1
SCHEMBL9646074 0.77 CCKBR (0.44) THRBLMNACYP3A4CYP2C9TSHR
SCHEMBL9558525 0.76 ALDH1A1 (0.43) LMNAALDH1A1CCKBRMMP1
SCHEMBL9559158 0.76 GAA (0.48) LMNAALDH1A1CCKBRMMP1
SCHEMBL9558853 0.75 ALDH1A1 (0.43) LMNAALDH1A1CCKBRMMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3151355-A None JP disclosed
EP-0508004-A1 Phenylsulfonylalkanoic acid compounds Kissei Pharmaceutical Co., Ltd. (JP) 1992-10-14 EP disclosed
US-5145869-A Treatment of irritable bowel syndrome, dyskinesia, pancreatist; hormone inhibitors KISSEI PHARMACEUTICAL CO., LTD. (JP) 1992-09-08 US disclosed
JP-H03151355-A PHENYLSULFONYLALKYLCARBOXYLIC ACID DERIVATIVE KISSEI PHARMACEUT CO LTD 1991-06-27 JP disclosed