SCHEMBL9656295

SCHEMBL9656295

O=C(O)CCCc1ccc(NS(=O)(=O)c2cccc(C(F)(F)F)c2)cn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.54
NR3C1 P04150 1/20 0.50
PGR P06401 1/20 0.50
AR P10275 1/20 0.50
ESR2 Q92731 1/20 0.50
HSD17B2 P37059 1/20 0.49
HDAC1 Q13547 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
SERPINE1 P05121 1/20 0.48
KMT2A Q03164 3/20 0.47
GAA P10253 2/20 0.47
MEN1 O00255 1/20 0.47
PIK3CB P42338 1/20 0.47
CA2 P00918 2/20 0.46
TRPV1 Q8NER1 1/20 0.45
CA1 P00915 1/20 0.45
MMP1 P03956 1/20 0.45
MMP2 P08253 1/20 0.45
MMP9 P14780 1/20 0.45
MMP8 P22894 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9654495 0.85 HDAC1 (0.52) HDAC1HDAC8KMT2AMEN1
SCHEMBL9656208 0.84 PGR (0.52) PGRHDAC1HDAC8
SCHEMBL9517143 0.84 TSHR (0.61) TSHRNR3C1PGRARESR2
SCHEMBL9657802 0.81 HDAC1 (0.53) HDAC1HDAC8KMT2AMEN1
SCHEMBL9656327 0.79 PTGDR2 (0.48) PGRHDAC1HDAC8KMT2AMEN1
SCHEMBL27630137 0.79 MEN1 (0.60) TSHRNR3C1PGRARESR2
SCHEMBL9656899 0.77 TBXAS1 (0.51) KMT2AMEN1
SCHEMBL9654550 0.77 IDO1 (0.49) ARHDAC1HDAC8KMT2AMEN1
SCHEMBL9656883 0.77 ALDH1A1 (0.60) KMT2AGAAMEN1CA2CA1
SCHEMBL10471236 0.76 FABP1 (0.47) HDAC1HDAC8KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0287270-B1 BIOLOGICALLY ACTIVE COMPOUNDS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1992-12-30 EP disclosed
US-4902698-A Benzenesulphonamidopyridyl compounds which are useful as thromboxane A.sub.2 SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1990-02-20 US disclosed
EP-0287270-A1 Biologically active compounds SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1988-10-19 EP disclosed