SCHEMBL9670261

SCHEMBL9670261

CS(=O)(=O)Nc1ccc([AsH]CC2CN(Cc3ccccc3)CCN2c2ccccc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 6/20 0.47
GRIN2B Q13224 2/20 0.39
POLB P06746 1/20 0.38
ACHE P22303 1/20 0.38
DRD2 P14416 1/20 0.38
ROCK2 O75116 3/20 0.38
NPC1 O15118 1/20 0.37
AR P10275 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9595403 0.85 ADRB1 (0.62) ADRB1GRIN2BPOLBACHEDRD2
SCHEMBL9595026 0.80 ADRB1 (0.66) ADRB1GRIN2BSMN1; SMN2
SCHEMBL9595783 0.77 ALDH1A1 (0.45) ADRB1GRIN2BPOLBROCK2NPC1
SCHEMBL8781020 0.72 DRD4 (0.60) ADRB1POLBDRD2
SCHEMBL9594552 0.69 SIGMAR1 (0.50) GRIN2BPOLBACHEDRD2
SCHEMBL25154608 0.68 DRD4 (0.46) GRIN2BSMN1; SMN2
SCHEMBL25154267 0.68 DRD4 (0.46) GRIN2BSMN1; SMN2
SCHEMBL14578035 0.67 ALDH1A1 (0.56) GRIN2BACHESMN1; SMN2
SCHEMBL18618573 0.67 SIGMAR1 (0.54)
SCHEMBL21455307 0.67 PKM (0.51) POLBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0491709-A1 2-SUBSTITUTED-1(4)-ARYL PIPERAZINES AND THE PROCESS FOR THEIR PREPARATION SCHERING AKTIENGESELLSCHAFT (DE) 1992-07-01 EP disclosed
WO-1991004250-A1 2-SUBSTITUTED-1(4)-ARYL PIPERAZINES AND THE PROCESS FOR THEIR PREPARATION SCHERING AKTIENGESELLSCHAFT BERLIN UND BERGKAMEN (DE) 1991-04-04 WO disclosed