SCHEMBL9673115

SCHEMBL9673115

BrCc1[c]ccc(-c2ccccc2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
MAPK1 P28482 2/20 0.38
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
TRPA1 O75762 1/20 0.34
TSHR P16473 1/20 0.34
MAOA P21397 1/20 0.34
NOTUM Q6P988 1/20 0.34
ALOX5 P09917 1/20 0.33
PTPN1 P18031 1/20 0.33
GSK3B P49841 1/20 0.33
ACMSD Q8TDX5 2/20 0.32
DHFR P00374 1/20 0.32
HNF4A P41235 1/20 0.32
MCL1 Q07820 1/20 0.32
AGXT P21549 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
MGLL Q99685 1/20 0.31
ERBB2 P04626 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1370479 0.80 ALDH1A1 (0.36) ALDH1A1MAPK1CRHBPCRHR2MAOA
SCHEMBL28489388 0.80 NOTUM (0.38) ALDH1A1CRHBPCRHR2TSHRMAOA
SCHEMBL27772757 0.80 TAAR1 (0.43) ALDH1A1MAPK1MAOANOTUMALOX5
SCHEMBL7877438 0.78 CALM1 (0.41) ALDH1A1TSHRMAOAPTPN1ACMSD
SCHEMBL6640494 0.77 TAAR1 (0.50) ALDH1A1TSHRKDM4EUSP2
SCHEMBL1372022 0.77 ALDH1A1 (0.39) ALDH1A1MAOAALOX5MCL1KDM4E
SCHEMBL533564 0.77 ALDH1A1 (0.42) ALDH1A1MAPK1CRHBPCRHR2MAOA
SCHEMBL8521841 0.76 PTGS2 (0.35) ALDH1A1MAPK1MAOAALOX5ACMSD
SCHEMBL29056142 0.75 ALDH1A1 (0.46) ALDH1A1MAPK1CRHBPCRHR2MAOA
SCHEMBL1370037 0.74 HSD11B1 (0.37) ALDH1A1TSHRMGLLKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519831-A1 N-Substituted heterocyclic derivatives, their preparation, and pharmaceutical compositions containing them SANOFI (FR) 1992-12-23 EP disclosed