SCHEMBL28489388

SCHEMBL28489388

OCc1[c]ccc(-c2ccccc2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.38
ALOX5 P09917 1/20 0.38
BACE1 P56817 1/20 0.37
CRHBP P24387 1/20 0.36
CRHR2 Q13324 1/20 0.36
ACMSD Q8TDX5 2/20 0.36
DHFR P00374 1/20 0.36
HNF4A P41235 1/20 0.36
MCL1 Q07820 1/20 0.36
ALDH1A1 P00352 2/20 0.36
MGLL Q99685 1/20 0.35
HDAC8 Q9BY41 2/20 0.35
PRKCI P41743 1/20 0.35
TSHR P16473 1/20 0.34
MAOA P21397 1/20 0.34
ESR2 Q92731 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
USP2 O75604 1/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9673115 0.80 ALDH1A1 (0.38) NOTUMALOX5CRHBPCRHR2ACMSD
SCHEMBL27772757 0.80 TAAR1 (0.43) NOTUMALOX5ALDH1A1MAOAKDM4E
SCHEMBL1370479 0.80 ALDH1A1 (0.36) ALOX5CRHBPCRHR2ACMSDDHFR
SCHEMBL7877438 0.78 CALM1 (0.41) ACMSDALDH1A1MGLLTSHRMAOA
SCHEMBL6640494 0.77 TAAR1 (0.50) ALDH1A1TSHRKDM4EUSP2HDAC2
SCHEMBL1372022 0.77 ALDH1A1 (0.39) ALOX5MCL1ALDH1A1MAOAKDM4E
SCHEMBL12479699 0.77 FFAR1 (0.51) ACMSDDHFRHNF4AMCL1ALDH1A1
SCHEMBL8521841 0.76 PTGS2 (0.35) ALOX5ACMSDDHFRHNF4AMCL1
SCHEMBL7390687 0.74 LMNA (0.39) ALDH1A1KDM4ELMNAHTT
SCHEMBL1370037 0.74 HSD11B1 (0.37) ALDH1A1MGLLTSHRKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112654610-A Pyrazole and imidazole compounds for inhibiting IL-17 and ROR gamma 里亚塔医药公司 2021-04-13 CN claimed
CN-112654610-A Pyrazole and imidazole compounds for inhibiting IL-17 and ROR gamma 里亚塔医药公司 2021-04-13 CN disclosed
CN-112105611-A Pharmaceutical combination comprising a Histone Deacetylase (HDAC) inhibitor and a TLR7 agonist and/or a TLR8 agonist for the treatment of cancer 4SC股份公司 2020-12-18 CN disclosed
CN-112055589-A Combination comprising an HDAC inhibitor, a LAG-3 inhibitor and a PD-1 inhibitor or a PD-L1 inhibitor for the treatment of cancer 4SC股份公司 2020-12-08 CN disclosed
CN-112004535-A Combination comprising an HDAC inhibitor and a CD137 agonist for cancer therapy 4SC股份公司 2020-11-27 CN disclosed