SCHEMBL9680343

SCHEMBL9680343

CCc1cc(CCc2nc3c(F)cccc3o2)c(=O)[nH]c1CO

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 2/20 0.41
PIK3CB P42338 2/20 0.41
DAGLA Q9Y4D2 1/20 0.34
HCAR2 Q8TDS4 1/20 0.34
TNKS O95271 2/20 0.33
PARP1 P09874 2/20 0.33
TNKS2 Q9H2K2 2/20 0.33
APLNR P35414 5/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 1/20 0.33
KMT2A Q03164 1/20 0.33
GLA P06280 2/20 0.32
TSHR P16473 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NPC1 O15118 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C19 P33261 1/20 0.31
RAB9A P51151 1/20 0.31
MCL1 Q07820 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9846133 0.86 PIK3CD (0.42) PIK3CDPIK3CBDAGLAHCAR2TNKS
SCHEMBL9680867 0.85 MEN1 (0.36) PIK3CDPIK3CBHCAR2TNKSPARP1
SCHEMBL9449230 0.83 MAPT (0.50) PIK3CDPIK3CBHCAR2APLNRMEN1
SCHEMBL9601892 0.77 ALDH1A1 (0.36) HCAR2APLNRALDH1A1MEN1HPGD
SCHEMBL9278111 0.75 PIK3CD (0.44) PIK3CDPIK3CBPARP1ALDH1A1MEN1
SCHEMBL9846224 0.73 PARP1 (0.37) PIK3CDPIK3CBTNKSPARP1TNKS2
SCHEMBL9846095 0.72 MAPT (0.50) PIK3CDPIK3CBAPLNRMEN1KMT2A
SCHEMBL9280614 0.71 PIK3CD (0.42) PIK3CDPIK3CBPARP1ALDH1A1MEN1
SCHEMBL9846101 0.70 ALDH1A1 (0.38) HCAR2TNKSPARP1TNKS2ALDH1A1
SCHEMBL9846186 0.70 MAPT (0.48) PIK3CDPIK3CBHCAR2APLNRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP claimed
EP-0481802-A1 Hydroxylated inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1992-04-22 EP disclosed