SCHEMBL9681249

SCHEMBL9681249

O=[N+]([O-])c1ccc2c(c1)c(N1CCNCC1)nn2-c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.48
HTR7 P34969 1/20 0.48
ADRB1 P08588 1/20 0.48
SIRT6 Q8N6T7 1/20 0.48
KHK P50053 2/20 0.46
CA9 Q16790 2/20 0.46
CA12 O43570 1/20 0.45
HTR3E A5X5Y0 1/20 0.45
HTR3B O95264 1/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
SLC6A4 P31645 1/20 0.45
CYP2C19 P33261 1/20 0.45
THPO P40225 1/20 0.45
HTR3A P46098 1/20 0.45
HTR3D Q70Z44 1/20 0.45
HTR3C Q8WXA8 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9682515 0.86 ADRB1 (0.57) HTR1AHTR7ADRB1SIRT6KHK
SCHEMBL9680678 0.80 KHK (0.51) HTR1AHTR7ADRB1KHKCA9
SCHEMBL9682532 0.80 KHK (0.51) HTR1AHTR7ADRB1KHKHTR3E
SCHEMBL2710715 0.79 KHK (0.54) ADRB1KHKHTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL9681346 0.78 KHK (0.53) ADRB1KHKHTR3EHTR3BHTR3A
SCHEMBL9683199 0.77 HTR1D (0.51) ADRB1KHKHTR3EHTR3BALDH1A1
SCHEMBL7114374 0.75 ALDH1A1 (0.52) CA9CA12ALDH1A1
SCHEMBL3649707 0.75 L3MBTL1 (0.50) CA9CA12ALDH1A1
SCHEMBL9681273 0.72 KHK (0.57) HTR1AHTR7ADRB1KHKHTR3E
SCHEMBL9680691 0.72 KHK (0.57) ADRB1KHKHTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed