SCHEMBL9681924

SCHEMBL9681924

C=CCN1CCN(c2nn(-c3ccccc3)c3ccccc23)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.47
HTR2C P28335 4/20 0.47
HTR3E A5X5Y0 2/20 0.47
HTR3B O95264 2/20 0.47
HTR3A P46098 2/20 0.47
HTR3D Q70Z44 2/20 0.47
HTR3C Q8WXA8 2/20 0.47
MAPT P10636 4/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CASP1 P29466 1/20 0.45
CYP2C19 P33261 1/20 0.45
CASP7 P55210 1/20 0.45
SMO Q99835 1/20 0.41
KHK P50053 2/20 0.41
PTGER1 P34995 1/20 0.41
LMNA P02545 3/20 0.40
DRD3 P35462 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9680620 0.99 HTR1A (0.47) HTR1AHTR2CHTR3EHTR3BHTR3A
SCHEMBL9681232 0.90 HTR1A (0.44) HTR1AHTR2CHTR3EHTR3BHTR3A
Bromide SCHEMBL9681411 0.89 HTR1A (0.44) HTR1AHTR2CHTR3EHTR3BHTR3A
SCHEMBL9682450 0.83 DRD4 (0.58) HTR1AHTR2CHTR3EHTR3BHTR3A
SCHEMBL9680636 0.82 SMO (0.50) MAPTSMOKHKPTGER1LMNA
SCHEMBL9680605 0.81 DRD2 (0.57) HTR1AHTR2CMAPTKHKLMNA
SCHEMBL9681250 0.81 HTR1A (0.60) HTR1AMAPTLMNAALDH1A1POLB
SCHEMBL9681419 0.81 KDM4E (0.49) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL9680621 0.80 KHK (0.44) MAPTCYP1A2CYP3A4CYP2D6SMO
SCHEMBL9682466 0.80 DRD3 (0.47) HTR1AHTR2CMAPTCYP2D6KHK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US disclosed
EP-0302423-A2 1-Phenyl-3-(1-piperazinyl)-1h-indazoles, a process and intermediates for their preparation, and the use thereof as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-02-08 EP disclosed