SCHEMBL9681232

SCHEMBL9681232

C=CCN1CCN(c2nn(-c3ccc(F)cc3)c3ccccc23)CC1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.44
HTR2C P28335 5/20 0.44
HTR3E A5X5Y0 3/20 0.44
HTR3B O95264 3/20 0.44
HTR3A P46098 3/20 0.44
HTR3D Q70Z44 3/20 0.44
HTR3C Q8WXA8 3/20 0.44
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C9 P11712 1/20 0.42
CASP1 P29466 1/20 0.42
CYP2C19 P33261 1/20 0.42
CASP7 P55210 1/20 0.42
SMO Q99835 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL9681411 0.99 HTR1A (0.44) HTR1AHTR2CHTR3EHTR3BHTR3A
SCHEMBL9681924 0.90 HTR1A (0.47) HTR1AHTR2CHTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL9680620 0.89 HTR1A (0.47) HTR1AHTR2CHTR3EHTR3BHTR3A
SCHEMBL9763064 0.84 KHK (0.51) LMNACYP1A2CYP3A4CYP2D6SMO
Hydrochloric Acid SCHEMBL9681944 0.83 KHK (0.50) LMNACYP1A2CYP3A4CYP2D6SMO
SCHEMBL9681952 0.81 LMNA (0.45) HTR1AHTR2CHTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL9680782 0.81 LMNA (0.44) HTR1AHTR2CHTR3EHTR3BHTR3A
SCHEMBL9681940 0.80 KHK (0.48) HTR1AHTR2CHTR3EHTR3BHTR3A
SCHEMBL9681305 0.78 KHK (0.47) HTR1AHTR2CHTR3AMAPT
SCHEMBL9680606 0.75 TP53 (0.45) LMNAMAPTSMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4999356-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-03-12 US claimed
US-5134236-A Analgesics, antidepressants, anticonvulsants HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-07-28 US disclosed