SCHEMBL9683346

SCHEMBL9683346

C=CCN1C2c3ccccc3C1c1sccc12

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PRCP P42785 3/20 0.38
OPRM1 P35372 1/20 0.35
CASP3 P42574 1/20 0.33
OPRD1 P41143 1/20 0.33
HHAT Q5VTY9 1/20 0.32
HTR1A P08908 2/20 0.32
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 2/20 0.31
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
KMT2A Q03164 1/20 0.31
HSD17B10 Q99714 1/20 0.31
ADRA1D P25100 1/20 0.30
ADRA1A P35348 1/20 0.30
ADRA1B P35368 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9683453 0.77 OPRM1 (0.35) OPRM1
SCHEMBL9684243 0.77 CHRM2 (0.37) ALDH1A1MAPTHPGDKMT2AHSD17B10
SCHEMBL9684281 0.76 OPRM1 (0.37) OPRM1
SCHEMBL9684167 0.75 ALDH1A1 (0.31) ALDH1A1HPGD
SCHEMBL9683465 0.74 CARM1 (0.33) OPRM1HTR1AKDM4EMEN1TSHR
SCHEMBL9684632 0.72 SLC6A2 (0.36) OPRM1HTR1AKDM4EMEN1TSHR
SCHEMBL9684133 0.72 CYP2D6 (0.38) OPRM1HTR1AALDH1A1KDM4EMEN1
SCHEMBL9683338 0.72 POLB (0.34) ALDH1A1KDM4EMEN1MAPTHPGD
SCHEMBL9682581 0.70 HTT (0.35) HHATKDM4EHPGD
SCHEMBL9684260 0.67 DUT (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0475187-A1 Naphthothiophenimines for treating neuronal disorders caused by ischemia BRISTOL-MYERS SQUIBB COMPANY (US) 1992-03-18 EP disclosed
US-5064831-A N-methyl-d-aspartate receptor antagonist BRISTOL-MYERS SQUIBB CO. (US) 1991-11-12 US disclosed