SCHEMBL9683458

SCHEMBL9683458

Nc1cc(F)ccc1NCc1ccc(Cl)c(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SSTR3 P32745 2/20 0.51
CYP2D6 P10635 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP1A2 P05177 1/20 0.49
SHMT2 P34897 1/20 0.43
ALDH1A1 P00352 1/20 0.41
HDAC3 O15379 1/20 0.40
NCOR1 O75376 1/20 0.40
CYP3A4 P08684 1/20 0.40
GAA P10253 1/20 0.40
FFAR1 O14842 1/20 0.40
CISD1 Q9NZ45 1/20 0.39
TSHR P16473 1/20 0.39
CD38 P28907 1/20 0.39
HDAC1 Q13547 1/20 0.39
PNMT P11086 1/20 0.39
TAAR1 Q96RJ0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681343 0.84 HDAC3 (0.44) SHMT2ALDH1A1HDAC3NCOR1GAA
SCHEMBL9683512 0.84 TP53 (0.46) SSTR3ALDH1A1GAAFFAR1TSHR
SCHEMBL16489601 0.82 ALDH1A1 (0.46) SSTR3CYP2D6CYP2C9CYP2C19ALDH1A1
SCHEMBL12658350 0.81 SHMT2 (0.48) SHMT2ALDH1A1HDAC3NCOR1HDAC1
SCHEMBL10507600 0.80 SSTR3 (0.51) SSTR3ALDH1A1GAAFFAR1CD38
SCHEMBL9681871 0.78 MAPT (0.43) SHMT2ALDH1A1HDAC3NCOR1HDAC1
SCHEMBL11569274 0.78 ALDH1A1 (0.49) ALDH1A1GAACISD1
SCHEMBL9683160 0.76 MAPT (0.54) SSTR3CYP2D6CYP2C9CYP2C19CYP1A2
SCHEMBL18768917 0.76 CYP1A2 (0.59) SSTR3CYP2D6CYP2C9CYP2C19CYP1A2
SCHEMBL9683331 0.75 MAP2K4 (0.52) GAAHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5128359-A Benzimidazole and azabenzimidazole derivatives which are thromboxane receptor antagonists, their methods of preparation LABORATOIRES UPSA (FR) 1992-07-07 US disclosed
US-5124336-A Cardiovascular disorders LABORATOIRES UPSA (FR) 1992-06-23 US disclosed
US-5021443-A Noval benzimidazole and azabenzimiazole derivatives which are thromboxane receptor antagonists, their methods of preparation and pharmaceutical compositions in which they are present LABORATOIRES UPSA (FR) 1991-06-04 US disclosed