SCHEMBL9683676

SCHEMBL9683676

CN1CC(Oc2ccccc2)C1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.56
SLC6A3 Q01959 2/20 0.56
HRH1 P35367 1/20 0.48
CARM1 Q86X55 1/20 0.47
PRMT6 Q96LA8 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CHRM3 P20309 2/20 0.47
NAAA Q02083 1/20 0.47
CHRM4 P08173 1/20 0.47
SLC6A4 P31645 2/20 0.46
USP30 Q70CQ3 2/20 0.42
CHRM2 P08172 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16707767 0.92 SLC6A2 (0.53) SLC6A2SLC6A3HRH1CARM1PRMT6
Sulfuric Acid SCHEMBL9596786 0.89 CHRM3 (0.47) SLC6A2SLC6A3CARM1PRMT6SMN1; SMN2
Maleic Acid SCHEMBL9682566 0.86 CHRM3 (0.49) SLC6A2SLC6A3HRH1SMN1; SMN2CHRM3
Fumaric Acid SCHEMBL9682573 0.86 CHRM3 (0.49) SLC6A2SLC6A3HRH1SMN1; SMN2CHRM3
SCHEMBL714763 0.86 SMN1; SMN2 (0.59) SLC6A2SLC6A3HRH1CARM1PRMT6
SCHEMBL10261345 0.86 SMN1; SMN2 (0.59) SLC6A2SLC6A3HRH1CARM1PRMT6
SCHEMBL10262302 0.86 SMN1; SMN2 (0.59) SLC6A2SLC6A3HRH1CARM1PRMT6
SCHEMBL21599178 0.82 SLC6A2 (0.45) SLC6A2SLC6A3HRH1CARM1PRMT6
SCHEMBL6585850 0.81 CHRM4 (0.54) SLC6A2SLC6A3CARM1PRMT6SMN1; SMN2
SCHEMBL20217571 0.81 HTR2C (0.46) SLC6A2SLC6A3SMN1; SMN2NAAAHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 49 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5130309-A Cardiovascular disorders A. H. ROBINS COMPANY, INCORPORATED (US) 1992-07-14 US claimed
WO-2023222850-A1 AMIDO HETEROAROMATIC COMPOUNDS USEFUL IN THE TREATMENT OF LIVER DISEASES ASTRAZENECA AB (SE) 2023-11-23 WO disclosed
EP-3262036-B1 THERAPEUTIC PYRIDAZINE COMPOUNDS AND USES THEREOF GENENTECH INC (US) 2023-09-13 EP disclosed
US-20230112485-A1 THERAPEUTIC COMPOUNDS GENENTECH, INC. (US) 2023-04-13 US disclosed
EP-3943490-A1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS Mission Therapeutics Limited (GB) 2022-01-26 EP disclosed
US-11066365-B2 1-cyano-pyrrolidine compounds as USP30 inhibitors MISSION THERAPEUTICS LIMITED (GB) 2021-07-20 US disclosed
EP-3277677-B9 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS MISSION THERAPEUTICS LTD (GB) 2021-07-14 EP disclosed
US-11053198-B2 1-cyano-pyrrolidine compounds as USP30 inhibitors MISSION THERAPEUTICS LIMITED (GB) 2021-07-06 US disclosed
EP-3842427-A1 1-CYANO-PYRROLIDINE COMPOUNDS AS USP30 INHIBITORS Mission Therapeutics Limited (GB) 2021-06-30 EP disclosed
US-11014912-B2 Cyanopyrrolidine derivatives with activity as inhibitors of USP30 MISSION THERAPEUTICS LIMITED (GB) 2021-05-25 US disclosed
US-20140243313-A1 TRICYCLIC COMPOUNDS USEFUL AS NEUROGENIC AND NEUROPROTECTIVE AGENTS INCEPTION ORION, INC. 2014-08-28 US disclosed
EP-2206707-B1 AZOLECARBOXAMIDE COMPOUND OR SALT THEREOF ASTELLAS PHARMA INC (JP) 2014-07-23 EP disclosed
US-8304547-B2 Azolecarboxamide compound or salt thereof ASTELLAS PHARMA INC. (JP) 2012-11-06 US disclosed
US-8304547-B2 Azolecarboxamide compound or salt thereof ASTELLAS PHARMA INC. (JP) 2012-11-06 US disclosed
US-20120028953-A1 Azetidine Derivatives VERNALIS (R&D) LTD. (GB) 2012-02-02 US disclosed
US-20110306587-A1 UNSATURATED NITROGEN HETEROCYCLIC COMPOUNDS USEFUL AS PDE10 INHIBITORS AMGEN INC. 2011-12-15 US disclosed
US-20100249088-A1 AZOLECARBOXAMIDE COMPOUND OR SALT THEREOF ASTELLAS PHARMA INC. (JP) 2010-09-30 US disclosed
EP-2206707-A1 AZOLECARBOXAMIDE COMPOUND OR SALT THEREOF Astellas Pharma Inc. (JP) 2010-07-14 EP disclosed
US-7494988-B2 Inhibitors of serine proteases, particularly hepatitis C virus NS3 protease VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-02-24 US disclosed
US-7494988-B2 Inhibitors of serine proteases, particularly hepatitis C virus NS3 protease VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-02-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11014912-B2 Cyanopyrrolidine derivatives with activity as inhibitors of USP30 USP30, USP39, USP28 SLC6A2 4696/4885SLC6A3 4618/4885HRH1 2856/4885
US-11066365-B2 1-cyano-pyrrolidine compounds as USP30 inhibitors USP30, USP20, USP10 SLC6A2 4669/4885SLC6A3 4448/4885HRH1 3070/4885
US-20140243313-A1 TRICYCLIC COMPOUNDS USEFUL AS NEUROGENIC AND NEUROPROTECTIVE AGENTS BDNF, GAP43, NLN SLC6A2 61/4885SLC6A3 89/4885HRH1 1301/4885
US-20230112485-A1 THERAPEUTIC COMPOUNDS BRDT, BRPF3, SNRPE SLC6A2 3813/4885SLC6A3 3416/4885HRH1 2718/4885
US-20120028953-A1 Azetidine Derivatives FAAH2, FAAH, APEH SLC6A2 1159/4885SLC6A3 792/4885HRH1 18/4885
US-11053198-B2 1-cyano-pyrrolidine compounds as USP30 inhibitors USP30, USP20, USP10 SLC6A2 4503/4885SLC6A3 4124/4885HRH1 3037/4885
US-20100249088-A1 AZOLECARBOXAMIDE COMPOUND OR SALT THEREOF TRPV1, FGFR3, GPR17 SLC6A2 1855/4885SLC6A3 1196/4885HRH1 578/4885
US-20110306587-A1 UNSATURATED NITROGEN HETEROCYCLIC COMPOUNDS USEFUL AS PDE10 INHIBITORS PDE10A, PDE2A, PDE3A SLC6A2 1990/4885SLC6A3 353/4885HRH1 3083/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.