SCHEMBL9686176

SCHEMBL9686176

CCNC(=O)Cc1cnc(N2CCN(Cc3ccccc3)CC2)nc1NCC

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.57
ACHE P22303 5/20 0.46
KDM4E B2RXH2 3/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
ALDH1A1 P00352 2/20 0.44
ALOX15 P16050 1/20 0.44
MDM2 Q00987 1/20 0.43
CHRM4 P08173 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9685068 0.83 TRPA1 (0.64) TRPA1ACHEKDM4EMAPTMAPK1
SCHEMBL9686751 0.80 TRPA1 (0.61) TRPA1KDM4EMAPTMAPK1NPSR1
SCHEMBL9685091 0.78 TRPA1 (0.59) TRPA1KDM4EMAPTMAPK1NPSR1
SCHEMBL9684409 0.78 TRPA1 (0.59) TRPA1KDM4EMAPTMAPK1NPSR1
SCHEMBL9686187 0.76 TRPA1 (0.52) TRPA1ACHEKDM4EMAPTMAPK1
SCHEMBL9685390 0.76 TRPA1 (0.60) TRPA1KDM4EHDAC6LMNAHTT
SCHEMBL9685239 0.76 TRPA1 (0.60) TRPA1KDM4EMAPTNPSR1HDAC6
SCHEMBL8812740 0.73 LMNA (0.52) TRPA1ACHEHDAC6LMNAHTT
SCHEMBL8812814 0.73 KDM4E (0.51) TRPA1ACHEKDM4EMAPTMAPK1
SCHEMBL8810744 0.72 HTT (0.46) TRPA1ACHEMAPTLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0188094-B1 QUINAZOLINE DERIVATIVES AND ANTIHYPERTENSIVE PREPARATIONS CONTAINING SAME AS EFFECTIVE COMPONENTS MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1992-03-18 EP disclosed
US-4734418-A Quinazoline compounds and antihypertensives MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1988-03-29 US disclosed
EP-0188094-A2 Quinazoline derivatives and antihypertensive preparations containing same as effective components MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1986-07-23 EP disclosed