SCHEMBL9686871

SCHEMBL9686871

CCn1cc(C#N)c2nc(N3CCNCC3)ncc2c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 18/20 0.43
CASP1 P29466 17/20 0.43
ALDH1A1 P00352 17/20 0.43
HSD17B10 Q99714 17/20 0.43
CASP7 P55210 16/20 0.43
HPGD P15428 12/20 0.43
CYP2C9 P11712 10/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
CYP3A4 P08684 12/20 0.40
TSHR P16473 6/20 0.40
CYP2C19 P33261 5/20 0.40
USP2 O75604 10/20 0.40
LMNA P02545 2/20 0.39
HIF1A Q16665 9/20 0.39
GLA P06280 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
TP53 P04637 1/20 0.38
MAPK1 P28482 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9685325 0.86 CYP1A2 (0.46) CYP1A2CASP1ALDH1A1HSD17B10CASP7
SCHEMBL9686741 0.81 CYP1A2 (0.41) CYP1A2CASP1ALDH1A1HSD17B10CASP7
SCHEMBL9686692 0.79 ABCC1 (0.41) CYP1A2CASP1ALDH1A1HSD17B10CASP7
SCHEMBL9686738 0.76 FNTA (0.44) ALDH1A1HSD17B10HPGDMEN1KMT2A
SCHEMBL9685229 0.74 USP19 (0.51) CYP1A2CASP1ALDH1A1HSD17B10CASP7
SCHEMBL10048250 0.70 CASP1 (0.57) CYP1A2CASP1ALDH1A1HSD17B10CASP7
SCHEMBL10678247 0.69 CASP1 (0.47) CYP1A2CASP1ALDH1A1HSD17B10CASP7
Pipemidic Acid SCHEMBL9935838 0.69 LMNA (0.80) CASP1ALDH1A1HSD17B10HPGDCYP2C9
Pipemidic Acid SCHEMBL675597 0.69 LMNA (0.80) CASP1ALDH1A1HSD17B10HPGDCYP2C9
Hydrochloric Acid SCHEMBL10508297 0.68 CASP1 (0.47) CYP1A2CASP1ALDH1A1HSD17B10CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0188094-B1 QUINAZOLINE DERIVATIVES AND ANTIHYPERTENSIVE PREPARATIONS CONTAINING SAME AS EFFECTIVE COMPONENTS MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1992-03-18 EP disclosed
US-4734418-A Quinazoline compounds and antihypertensives MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1988-03-29 US disclosed
EP-0188094-A2 Quinazoline derivatives and antihypertensive preparations containing same as effective components MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1986-07-23 EP disclosed