SCHEMBL9686692

SCHEMBL9686692

CCn1cc(C#N)c2nc(N3CCN(OCc4ccccc4)CC3)ncc2c1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 9/20 0.41
ALDH1A1 P00352 4/20 0.36
HSD17B10 Q99714 4/20 0.36
CASP1 P29466 3/20 0.36
USP2 O75604 3/20 0.36
CYP1A2 P05177 3/20 0.36
TSHR P16473 3/20 0.36
HPGD P15428 2/20 0.36
CASP7 P55210 2/20 0.36
KDM4E B2RXH2 3/20 0.36
MAPK1 P28482 1/20 0.36
LMNA P02545 2/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP3A4 P08684 2/20 0.35
ABCB1 P08183 1/20 0.35
TP53 P04637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9686738 0.86 FNTA (0.44) ABCC1ALDH1A1HSD17B10HPGDKDM4E
SCHEMBL9686871 0.79 CYP1A2 (0.43) ALDH1A1HSD17B10CASP1USP2CYP1A2
SCHEMBL9686660 0.74 HTT (0.48) ALDH1A1HSD17B10CASP1USP2TSHR
SCHEMBL9684377 0.71 PTPN11 (0.42) ALDH1A1HSD17B10CASP1HPGDKDM4E
SCHEMBL9686146 0.70 HTT (0.46) ALDH1A1HSD17B10CASP1USP2TSHR
SCHEMBL9685325 0.66 CYP1A2 (0.46) ALDH1A1HSD17B10CASP1USP2CYP1A2
SCHEMBL9684556 0.65 LMNA (0.51) ALDH1A1HSD17B10CASP1TSHRHPGD
SCHEMBL9686858 0.63 HTR3A (0.55) ALDH1A1HSD17B10CASP1USP2CYP1A2
SCHEMBL9686741 0.62 CYP1A2 (0.41) ALDH1A1HSD17B10CASP1USP2CYP1A2
SCHEMBL3521025 0.60 MAOB (0.49) ALDH1A1HSD17B10CASP1CYP1A2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0188094-B1 QUINAZOLINE DERIVATIVES AND ANTIHYPERTENSIVE PREPARATIONS CONTAINING SAME AS EFFECTIVE COMPONENTS MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1992-03-18 EP disclosed
US-4734418-A Quinazoline compounds and antihypertensives MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1988-03-29 US disclosed
EP-0188094-A2 Quinazoline derivatives and antihypertensive preparations containing same as effective components MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1986-07-23 EP disclosed