SCHEMBL9689140

SCHEMBL9689140

COc1ccc(CCN(C)C)c2[nH]cnc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.47
HTR1A P08908 3/20 0.45
ABL1 P00519 1/20 0.40
RAD52 P43351 1/20 0.40
RIN1 Q13671 1/20 0.40
HTR2A P28223 2/20 0.40
AOC3 Q16853 1/20 0.39
HTR7 P34969 2/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38
HTR2C P28335 1/20 0.38
HTR1E P28566 1/20 0.38
HTR1F P30939 1/20 0.38
HTR2B P41595 1/20 0.38
HTR3A P46098 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9689134 0.89 HTR6 (0.50) HTR6HTR1AABL1RAD52RIN1
SCHEMBL9689677 0.85 SIGMAR1 (0.40)
SCHEMBL9689133 0.79 HTR1A (0.46) HTR6HTR1AHTR2AHTR7HTR1D
SCHEMBL9687954 0.76 HTR6 (0.43) HTR6HTR1AHTR2AAOC3HTR7
SCHEMBL2272157 0.76 ABL1 (0.53) ABL1RAD52RIN1
SCHEMBL9689684 0.75 NOS1 (0.43) HTR6HTR1AHTR2AAOC3NOS1
SCHEMBL9689665 0.74 SIGMAR1 (0.40)
SCHEMBL9689122 0.74 HTR1A (0.46) HTR6HTR1AHTR2AHTR7HTR1D
SCHEMBL10409117 0.72 PDE4B (0.42) HTR6HTR1AHTR2AAOC3NOS1
SCHEMBL9689621 0.71 HTR6 (0.47) HTR6HTR1AHTR2AAOC3HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0189473-B1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1992-05-27 EP disclosed
US-4958026-A HYPOTENSIVE AGENTS SCHERING AKTIENGESLLSCHAFT (DE) 1990-09-18 US disclosed