SCHEMBL9689534

SCHEMBL9689534

COC(=O)OC1=C(C)NC(C)=C(OC(=O)O)C1c1ccccc1OCc1cccc(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 1/20 0.44
SLC1A5 Q15758 1/20 0.44
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MRGPRX4 Q96LA9 2/20 0.42
NR4A2 P43354 2/20 0.41
MAOB P27338 4/20 0.41
PPIA P62937 1/20 0.40
CACNA1F O60840 1/20 0.40
CACNA1D Q01668 1/20 0.40
CACNA1S Q13698 1/20 0.40
CACNA1C Q13936 1/20 0.40
PTGER1 P34995 1/20 0.40
KIFC1 Q9BW19 1/20 0.39
SLC26A3 P40879 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10814008 0.95 FFAR4 (0.48) FFAR4SLC1A5ALDH1A1GAAL3MBTL1
SCHEMBL9689636 0.92 CACNA1F (0.45) FFAR4SLC1A5ALDH1A1GAAL3MBTL1
SCHEMBL11169187 0.90 FFAR4 (0.41) FFAR4SLC1A5ALDH1A1GAAL3MBTL1
SCHEMBL10646682 0.88 SMYD3 (0.43) FFAR4SLC1A5ALDH1A1GAAL3MBTL1
SCHEMBL9691796 0.88 HTR6 (0.43) GAAL3MBTL1MRGPRX4NR4A2MAOB
SCHEMBL9691359 0.88 POLB (0.44) ALDH1A1GAAL3MBTL1
SCHEMBL10649923 0.88 L3MBTL1 (0.39) FFAR4SLC1A5ALDH1A1GAAL3MBTL1
SCHEMBL9691807 0.86 SLC1A5 (0.44) SLC1A5MRGPRX4
SCHEMBL10914095 0.85 POLB (0.46) ALDH1A1GAAL3MBTL1
SCHEMBL9691625 0.84 NR1I2 (0.42) SLC1A5ALDH1A1GAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed
EP-0288758-B1 DIHYDROPYRIDINAMIDES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN MEDICINES BAYER AG (DE) 1991-08-14 EP disclosed
EP-0071819-A1 Dihydropyridines with a positive inotropic activity, their use in pharmaceutical preparations, and processes for their preparation BAYER AG (DE) 1983-02-16 EP disclosed