SCHEMBL9689684

SCHEMBL9689684

COc1ccc(CCN(C)C)c2[nH]c(N)nc12

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 3/20 0.43
HTR6 P50406 2/20 0.42
AOC3 Q16853 3/20 0.40
HTR1A P08908 2/20 0.40
NOS3 P29474 1/20 0.40
PNP P00491 1/20 0.39
HTR2A P28223 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9689679 0.89 HTR6 (0.45) NOS1HTR6AOC3HTR1ANOS3
SCHEMBL9687954 0.85 HTR6 (0.43) NOS1HTR6AOC3HTR1ANOS3
SCHEMBL9688843 0.81 HTR1A (0.41) HTR6HTR1APNPHTR2A
SCHEMBL10409117 0.81 PDE4B (0.42) NOS1HTR6AOC3HTR1ANOS3
SCHEMBL9689985 0.80 HTR6 (0.39) NOS1HTR6AOC3HTR1ANOS3
SCHEMBL5924181 0.77 NQO2 (0.42) PNP
SCHEMBL9688833 0.75 HTR1A (0.41) HTR6HTR1APNPHTR2A
SCHEMBL9689140 0.75 HTR6 (0.47) NOS1HTR6AOC3HTR1AHTR2A
SCHEMBL9687943 0.74 HTR6 (0.46) NOS1HTR6AOC3HTR1ANOS3
SCHEMBL20795146 0.72 NQO2 (0.46) PNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0189473-B1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1992-05-27 EP disclosed
US-4958026-A HYPOTENSIVE AGENTS SCHERING AKTIENGESLLSCHAFT (DE) 1990-09-18 US disclosed