SCHEMBL9688833

SCHEMBL9688833

CN(C)CCc1ccc(O)c2[nH]c(N)nc12

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.41
HTR2A P28223 5/20 0.40
HTR2C P28335 4/20 0.37
HTR2B P41595 3/20 0.37
HTR7 P34969 2/20 0.37
DRD1 P21728 1/20 0.37
HTR1D P28221 1/20 0.37
HTR1B P28222 1/20 0.37
HTR1E P28566 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA2B P29275 1/20 0.37
DRD3 P35462 1/20 0.37
HTR5A P47898 1/20 0.37
HTR6 P50406 1/20 0.37
PNP P00491 2/20 0.36
SLC6A4 P31645 1/20 0.34
ADRB2 P07550 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9688843 0.89 HTR1A (0.41) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL9688933 0.84 ADRB2 (0.47) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL9689679 0.81 HTR6 (0.45) HTR1AHTR2AHTR6PNP
SCHEMBL9688999 0.80 HTR1A (0.41) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL9687965 0.79 HTR1A (0.38) HTR1AHTR2AHTR2CHTR2B
SCHEMBL9689684 0.75 NOS1 (0.43) HTR1AHTR2AHTR6PNP
SCHEMBL7993998 0.74 NUDT1 (0.42) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL9689808 0.74 HTR1A (0.43) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL9689122 0.74 HTR1A (0.46) HTR1AHTR2AHTR2CHTR2BHTR7
SCHEMBL9688945 0.72 ADRB2 (0.47) HTR1AHTR2AHTR2CHTR2BHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0189473-B1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1992-05-27 EP disclosed
US-4958026-A HYPOTENSIVE AGENTS SCHERING AKTIENGESLLSCHAFT (DE) 1990-09-18 US disclosed
EP-0189473-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS. SCHERING AG (DE) 1986-08-06 EP disclosed
WO-1986001204-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1986-02-27 WO disclosed