SCHEMBL9689688

SCHEMBL9689688

COc1ccc(CCN)c2c(=O)[nH][nH]c12

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.44
TAAR1 Q96RJ0 3/20 0.44
ADRA1A P35348 1/20 0.44
NEK1 Q96PY6 3/20 0.39
KDM4E B2RXH2 1/20 0.39
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9688657 0.76 DRD2 (0.44) TAAR1NEK1KDM4E
SCHEMBL9688896 0.75 HTR2A (0.47) HTR2ATAAR1ADRA1AKDM4EATM
SCHEMBL9688747 0.74 ALDH1A1 (0.51) KDM4E
SCHEMBL1190039 0.74 ADRB2 (0.44) HTR2ATAAR1ADRA1ANEK1
Hydrochloric Acid SCHEMBL1190213 0.72 ADRB2 (0.43) HTR2ATAAR1ADRA1ANEK1
SCHEMBL7281232 0.72 HTR2A (0.50) HTR2ATAAR1ADRA1ANEK1KDM4E
SCHEMBL9689779 0.71 HTR2A (0.43) HTR2ATAAR1ADRA1AKDM4EATM
SCHEMBL24498666 0.69 HTR2A (0.57) HTR2ATAAR1ADRA1A
SCHEMBL11816292 0.68 TAAR1 (0.58) HTR2ATAAR1ADRA1A
SCHEMBL8303296 0.67 TAAR1 (0.52) HTR2ATAAR1ADRA1AKDM4EATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0189473-B1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1992-05-27 EP disclosed
US-4958026-A HYPOTENSIVE AGENTS SCHERING AKTIENGESLLSCHAFT (DE) 1990-09-18 US disclosed
EP-0189473-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS. SCHERING AG (DE) 1986-08-06 EP disclosed
WO-1986001204-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1986-02-27 WO disclosed