SCHEMBL9689825

SCHEMBL9689825

CN1CCC(Nc2nc3cccnc3[nH]2)C1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.47
DBF4 Q9UBU7 1/20 0.47
CHEK2 O96017 1/20 0.42
RET P07949 1/20 0.42
KAT2B Q92831 1/20 0.40
KCNH2 Q12809 2/20 0.40
ERN1 O75460 1/20 0.39
MAPK10 P53779 1/20 0.39
DYRK1A Q13627 2/20 0.39
DYRK1B Q9Y463 2/20 0.39
SSTR4 P31391 3/20 0.38
HRH4 Q9H3N8 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
JAK2 O60674 4/20 0.37
JAK3 P52333 4/20 0.37
BRD4 O60885 1/20 0.37
ATAD2 Q6PL18 1/20 0.37
SSTR1 P30872 1/20 0.37
PIM1 P11309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9534992 0.92 CDC7 (0.54) CDC7DBF4RETKCNH2DYRK1A
Hydrochloric Acid SCHEMBL9535340 0.91 CDC7 (0.53) CDC7DBF4RETKCNH2DYRK1A
SCHEMBL27505138 0.78 JAK3 (0.43) CDC7DBF4KCNH2HRH4HRH3
SCHEMBL9044459 0.77 PTPN11 (0.48) CDC7DBF4HRH3BRD4ATAD2
SCHEMBL8135558 0.76 KCNH2 (0.45) CDC7DBF4RETKCNH2HRH3
SCHEMBL9687566 0.76 KCNH2 (0.42) CDC7DBF4KCNH2
Hydrochloric Acid SCHEMBL9535454 0.75 KCNH2 (0.51) CDC7DBF4KCNH2HRH3
SCHEMBL5054675 0.75 NOS2 (0.62) JAK2JAK3
SCHEMBL9689165 0.75 MKNK1 (0.45) CHEK2BRD4ATAD2
SCHEMBL9535712 0.74 KCNH2 (0.75) KCNH2HRH4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0297661-B1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-16 EP disclosed