SCHEMBL9689951

SCHEMBL9689951

COc1ccc2cc(-c3nnnn3C(C)C(=O)O)sc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.41
PPARA Q07869 3/20 0.39
PTGS2 P35354 3/20 0.39
AKR1C3 P42330 3/20 0.39
AKR1C2 P52895 3/20 0.39
PTGS1 P23219 2/20 0.39
CYP1A2 P05177 2/20 0.39
CDC42 P60953 1/20 0.39
RAC1 P63000 1/20 0.39
TSHR P16473 1/20 0.39
SLC22A6 Q4U2R8 1/20 0.39
NPC1 O15118 4/20 0.38
RAB9A P51151 4/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPT P10636 2/20 0.38
ATAD2 Q6PL18 1/20 0.38
CA2 P00918 1/20 0.38
SCD O00767 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9690025 0.91 PPARA (0.42) TDP1PPARAPTGS2AKR1C3AKR1C2
SCHEMBL9690648 0.87 NPSR1 (0.38) PPARATSHRMAPTSCD
SCHEMBL9688900 0.83 KDM4E (0.41) PTGS2PTGS1CYP1A2RAB9AKDM4E
SCHEMBL9689963 0.77 HDAC3 (0.43) NPC1RAB9AKDM4EMAPTCA2
SCHEMBL9689940 0.77 TDP1 (0.40) TDP1PPARAPTGS2AKR1C3AKR1C2
SCHEMBL9689398 0.72 TDP1 (0.41) TDP1PTGS2AKR1C3AKR1C2PTGS1
SCHEMBL9689396 0.71 KDM4E (0.49) TDP1KDM4EMAPTCA2MEN1
SCHEMBL3554931 0.69 KDM4E (0.56) TSHRNPC1RAB9AKDM4EMAPT
SCHEMBL9688521 0.68 SIGMAR1 (0.38) TDP1CYP1A2RAB9AKDM4EMAPT
SCHEMBL12871087 0.66 HDAC6 (0.56) CYP1A2TSHRNPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0506011-A1 Tetrazoleacetic acid derivatives having aldose reductase inhibitory activity Wakamoto Pharmaceutical Co., Ltd. (JP) 1992-09-30 EP disclosed