SCHEMBL9690877

SCHEMBL9690877

COC(=O)OC1=C(C)NC(C)=C(OC(=O)O)C1c1ccccc1OCc1ccc(Cl)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 2/20 0.43
FFAR1 O14842 3/20 0.40
TACR1 P25103 4/20 0.40
PTPRC P08575 1/20 0.39
PTPN1 P18031 1/20 0.39
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
NR1I2 O75469 1/20 0.37
HTR1A P08908 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
CARM1 Q86X55 1/20 0.37
PRMT1 Q99873 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10815688 0.94 HTR6 (0.47) HTR6FFAR1TACR1PTPRCPTPN1
SCHEMBL10649783 0.91 HTR6 (0.41) HTR6FFAR1TACR1PTPRCPTPN1
SCHEMBL9691359 0.88 POLB (0.44) KDM4EGAAMAPTNR1I2HTR1A
SCHEMBL10646848 0.88 HTR6 (0.43) HTR6FFAR1TACR1KDM4EGAA
SCHEMBL9691648 0.88 TP53 (0.41) KDM4EGAANPC1MAPTRAB9A
SCHEMBL9691625 0.87 NR1I2 (0.42) KDM4EGAAMAPTRAB9ANR1I2
SCHEMBL9690850 0.87 GAA (0.40) FFAR1TACR1KDM4EGAAMAPT
SCHEMBL9689430 0.86 ALDH1A1 (0.43) KDM4EGAAMAPTNR1I2SLC6A3
SCHEMBL9690847 0.86 FABP4 (0.45) FFAR1KDM4EGAANR1I2
SCHEMBL9691807 0.85 SLC1A5 (0.44) FFAR1KDM4EMAPTHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed
EP-0288758-A2 Dihydropyridinamides, process for their preparation and their use in medicines BAYER AG (DE) 1988-11-02 EP disclosed