SCHEMBL9692045

SCHEMBL9692045

COC(=O)C1=CCCN(CCC2CCOc3ccccc32)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.50
LMNA P02545 2/20 0.43
CHRM2 P08172 1/20 0.43
CHRM4 P08173 1/20 0.43
CHRM5 P08912 1/20 0.43
THRB P10828 1/20 0.43
CHRM1 P11229 1/20 0.43
CHRM3 P20309 1/20 0.43
BLM P54132 2/20 0.42
MCOLN3 Q8TDD5 1/20 0.42
OPRK1 P41145 1/20 0.40
HTR2A P28223 5/20 0.37
DRD2 P14416 4/20 0.37
DRD3 P35462 4/20 0.37
PTGDR2 Q9Y5Y4 2/20 0.36
HTR2C P28335 1/20 0.36
HRH1 P35367 1/20 0.36
HTR2B P41595 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9825506 0.88 SLC6A1 (0.47) KCNH2LMNABLMKDM4EALDH1A1
SCHEMBL9824935 0.84 KCNH2 (0.48) KCNH2HTR2ADRD2DRD3PTGDR2
SCHEMBL10395490 0.83 LMNA (0.46) LMNACHRM2CHRM4CHRM5THRB
Hydrochloric Acid SCHEMBL10394912 0.82 LMNA (0.45) LMNACHRM2CHRM4CHRM5THRB
SCHEMBL10685083 0.81 KCNH2 (0.52) KCNH2
SCHEMBL9692552 0.78 HTT (0.47) LMNACHRM2CHRM4CHRM5THRB
Hydrochloric Acid SCHEMBL9692396 0.78 HTT (0.46) LMNACHRM2CHRM4CHRM5THRB
SCHEMBL9692507 0.76 MALT1 (0.43) KCNH2LMNACHRM2CHRM4CHRM5
Hydrochloric Acid SCHEMBL9692497 0.75 MALT1 (0.42) KCNH2LMNACHRM2CHRM4CHRM5
SCHEMBL9824929 0.75 KCNH2 (0.49) KCNH2HTR2ADRD2DRD3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0252005-B1 HYDROGENATED 1-BENZOOXACYCLOALKYL-PYRIDINE CARBOXYLIC-ACID COMPOUNDS CIBA-GEIGY AG (CH) 1991-07-10 EP claimed
US-5112855-A Nootropic Agents CIBA-GEIGY CORPORATION (US) 1992-05-12 US disclosed
US-4957928-A NOOTROPIC AGENTS, COGNITION ACTIVATORS CIBA-GEIGY CORPORATION (US) 1990-09-18 US disclosed