SCHEMBL9824929

SCHEMBL9824929

COC(=O)OC1CCCN(CCC2CCOc3ccccc32)C1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.49
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP1A2 P05177 1/20 0.42
KDM4E B2RXH2 1/20 0.40
BCHE P06276 4/20 0.39
MAOB P27338 2/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
HTT P42858 1/20 0.38
DRD2 P14416 1/20 0.37
HTR2A P28223 1/20 0.37
DRD3 P35462 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9690362 0.78 ALDH1A1 (0.57) KDM4EMEN1KMT2ADRD2HTR2A
SCHEMBL9824935 0.78 KCNH2 (0.48) KCNH2DRD2HTR2ADRD3
SCHEMBL9825802 0.78 MALT1 (0.42) CYP3A4CYP2D6CYP1A2BCHEMAOB
SCHEMBL19852411 0.77 KCNH2 (0.46) KCNH2HTR2A
SCHEMBL19852525 0.77 KCNH2 (0.46) KCNH2HTR2A
SCHEMBL9692045 0.75 KCNH2 (0.50) KCNH2CYP2D6CYP1A2KDM4EKMT2A
SCHEMBL9339570 0.75 DRD2 (0.59) KCNH2DRD2HTR2ADRD3
SCHEMBL9825234 0.73 ADRA2A (0.55) DRD2
Hydrochloric Acid SCHEMBL9824882 0.72 ADRA2A (0.54) CYP2D6MEN1KMT2ADRD2
SCHEMBL10407828 0.71 DRD2 (0.48) KCNH2CYP3A4CYP1A2KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0252005-B1 HYDROGENATED 1-BENZOOXACYCLOALKYL-PYRIDINE CARBOXYLIC-ACID COMPOUNDS CIBA-GEIGY AG (CH) 1991-07-10 EP disclosed
EP-0252005-A1 Hydrogenated 1-benzooxacycloalkyl-pyridine carboxylic-acid compounds CIBA-GEIGY AG (CH) 1988-01-07 EP disclosed