SCHEMBL9697261

SCHEMBL9697261

CCC(NC(=O)OCc1ccccc1)P(=O)(O)CC(CCc1ccc2ccccc2c1)C(=O)OC

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP8 P22894 3/20 0.55
MMP14 P50281 3/20 0.55
MMP2 P08253 2/20 0.55
MMP7 P09237 2/20 0.55
MMP9 P14780 2/20 0.55
ACE2 Q9BYF1 1/20 0.51
ECE1 P42892 13/20 0.50
MME P08473 12/20 0.50
F2 P00734 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9698581 0.91 ACE2 (0.58) MMP8MMP14ACE2ECE1MME
SCHEMBL9715129 0.86 ACE2 (0.50) MMP8MMP14MMP2MMP7MMP9
SCHEMBL9715090 0.85 MMP8 (0.64) MMP8MMP14MMP2MMP9ACE2
SCHEMBL9715281 0.84 ACE2 (0.62) ACE2ECE1MME
SCHEMBL9697199 0.83 ACE2 (0.70) MMP8MMP14ACE2ECE1MME
SCHEMBL9715088 0.82 ECE1 (0.60) MMP8MMP14MMP2MMP9ACE2
SCHEMBL9715136 0.81 ACE2 (0.69) ACE2ECE1MME
SCHEMBL9698508 0.80 MMP8 (0.59) MMP8MMP14MMP2MMP9ACE2
SCHEMBL23881756 0.77 CASP1 (0.55) MMP8MMP14MMP2MMP7MMP9
SCHEMBL6928745 0.77 ECE1 (0.77) MMP8MMP14ACE2ECE1MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5143908-A Carboxylic acids containing amino and phosphinyl groups MERCK & CO., INC. (US) 1992-09-01 US disclosed
US-5099063-A 3-(1-aminoalkylphosphinyl)-(2-substituted)propionic acids MERCK & CO., INC. (US) 1992-03-24 US disclosed
EP-0266978-A2 Novel antibacterial agents and potentiators of carbapenem antibiotics MERCK & CO. INC. (US) 1988-05-11 EP disclosed
US-4715994-A PHOSPHINIC ACID DERIVATIVES MERCK & CO., INC. (US) 1987-12-29 US disclosed