SCHEMBL9728617

SCHEMBL9728617

COc1cccc2c1OCC(CN1CCSCC1)N2N

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.41
HTR1A P08908 3/20 0.41
ADRA1D P25100 3/20 0.41
ADRA1B P35368 3/20 0.41
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HTR7 P34969 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10378979 0.93 ADRA1A (0.38) ADRA1AHTR1AADRA1DADRA1BADRA2A
SCHEMBL9700351 0.90 ADRA2A (0.41) ADRA1AHTR1AADRA1DADRA1BADRA2A
SCHEMBL9701613 0.90 ADRA2A (0.41) ADRA1AHTR1AADRA1DADRA1BADRA2A
SCHEMBL9699337 0.87 ADRA2A (0.42) ADRA1AHTR1AADRA1DADRA1BADRA2A
SCHEMBL9699344 0.84 ADRA1A (0.42) ADRA1AHTR1AADRA1DADRA1BADRA2A
SCHEMBL9699287 0.83 HTR7 (0.40) ADRA1AHTR1AADRA1DADRA1BADRA2A
SCHEMBL9699340 0.82 CYP2A13 (0.39)
SCHEMBL9700158 0.80 HTR2A (0.38) ADRA1AHTR1AADRA1DADRA1BADRA2A
SCHEMBL10471313 0.80 ADRA2A (0.37) ADRA1AHTR1AADRA1DADRA1BADRA2A
SCHEMBL9700327 0.77 ADRA1D (0.38) ADRA1AHTR1AADRA1DADRA1BADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed