SCHEMBL9700309

SCHEMBL9700309

NCC1COc2c(Cl)cccc2N1N=O

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.38
CA2 P00918 1/20 0.34
HTR2A P28223 3/20 0.33
HTR2C P28335 3/20 0.33
HTR2B P41595 3/20 0.33
GAA P10253 2/20 0.32
RIPK1 Q13546 1/20 0.32
AADAT Q8N5Z0 1/20 0.31
PTPN11 Q06124 1/20 0.31
ADRA1D P25100 1/20 0.30
ADRA1A P35348 1/20 0.30
ADRA1B P35368 1/20 0.30
AKT1 P31749 1/20 0.30
HTR6 P50406 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9699339 0.83 NOTUM (0.39) NOTUMCA2GAARIPK1ADRA1D
SCHEMBL9699310 0.82 NOTUM (0.38) NOTUMADRA1DADRA1AADRA1B
SCHEMBL9699297 0.82 NOTUM (0.38) NOTUMADRA1DADRA1AADRA1B
SCHEMBL9699269 0.81 NOTUM (0.38) NOTUMCA2HTR2AHTR2CHTR2B
SCHEMBL9699348 0.81 NOTUM (0.39) NOTUMCA2GAARIPK1AADAT
SCHEMBL9701449 0.79 DRD2 (0.41) NOTUMHTR2AHTR2CHTR6
SCHEMBL9700270 0.79 CYP2A13 (0.37) NOTUM
SCHEMBL9701406 0.78 SMN1; SMN2 (0.37) CA2GAAADRA1A
SCHEMBL9700406 0.75 ADRB1 (0.38) NOTUMHTR2AHTR2CHTR2BHTR6
SCHEMBL9700400 0.75 HTR2A (0.34) NOTUMHTR2AHTR2CHTR2BHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed