SCHEMBL9699339

SCHEMBL9699339

CNCC1COc2c(Cl)cccc2N1N=O

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.39
RIPK1 Q13546 1/20 0.36
CA2 P00918 1/20 0.34
SLC6A4 P31645 3/20 0.33
CYP2D6 P10635 2/20 0.33
SLC6A2 P23975 2/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
AQP1 P29972 1/20 0.33
XIAP P98170 2/20 0.31
GAA P10253 1/20 0.30
DRD2 P14416 1/20 0.30
DRD3 P35462 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701394 0.84 ADRA1A (0.36) ADRA1DADRA1AADRA1BXIAPDRD2
SCHEMBL9700309 0.83 NOTUM (0.38) NOTUMRIPK1CA2ADRA1DADRA1A
SCHEMBL9700368 0.82 NOTUM (0.37) NOTUMRIPK1CA2SLC6A4CYP2D6
SCHEMBL9699310 0.79 NOTUM (0.38) NOTUMADRA1DADRA1AADRA1BDRD2
SCHEMBL9699297 0.79 NOTUM (0.38) NOTUMADRA1DADRA1AADRA1BDRD2
SCHEMBL9701449 0.78 DRD2 (0.41) NOTUMDRD2DRD3
SCHEMBL9700270 0.76 CYP2A13 (0.37) NOTUMDRD2DRD3
SCHEMBL9699348 0.75 NOTUM (0.39) NOTUMRIPK1CA2CYP2D6GAA
SCHEMBL9700406 0.72 ADRB1 (0.38) NOTUMCYP2D6DRD2DRD3
SCHEMBL9700400 0.72 HTR2A (0.34) NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed