SCHEMBL9700481

SCHEMBL9700481

NCC1CN(N)c2ccccc2O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 4/20 0.39
ADRA2A P08913 2/20 0.37
ADRA1A P35348 2/20 0.37
HTR1A P08908 1/20 0.37
DRD1 P21728 1/20 0.37
TBXA2R P21731 1/20 0.37
SLC6A2 P23975 1/20 0.37
DRD3 P35462 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
ADRA1D P25100 1/20 0.37
ADRA1B P35368 1/20 0.37
SCN1A P35498 1/20 0.37
SCN2A Q99250 1/20 0.37
SCN3A Q9NY46 1/20 0.37
SIRT1 Q96EB6 3/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HRH1 P35367 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9151791 0.84 HTR1A (0.40) CA2ADRA2AADRA1AHTR1ADRD1
SCHEMBL9153836 0.81 HTT (0.38) CA2ADRA2AADRA1AHTR1ADRD1
SCHEMBL2685298 0.81 CASR (0.49) HTR1ASIRT1SIRT2
SCHEMBL9699321 0.80 HTR6 (0.43) CA2ADRA2AADRA1AHTR1ADRD3
SCHEMBL9155416 0.79 HTT (0.46) SIRT1SIRT2
SCHEMBL9701487 0.79 ADRA2A (0.56) ADRA2AADRA1AHTR1AADRA2BADRA2C
SCHEMBL9701550 0.79 ADRA2A (0.60) ADRA2AADRA1AHTR1AADRA2BADRA2C
SCHEMBL9529252 0.78 CASR (0.50) ADRA1AHTR1AADRA1DADRA1B
SCHEMBL11805714 0.78 GRM2 (0.51)
SCHEMBL9699225 0.78 HTR2A (0.42) CA2SIRT1HTR2AHTR2CHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed