SCHEMBL9700639

SCHEMBL9700639

CC(C)C(C)(C)[Si](C)(C)OCCc1ccc(CCCC(CO)(CNC(=O)O)c2ccccc2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
HTT P42858 1/20 0.35
NAAA Q02083 1/20 0.33
KMT2A Q03164 2/20 0.33
HPGD P15428 2/20 0.33
EDNRB P24530 5/20 0.33
EDNRA P25101 5/20 0.33
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
POLB P06746 1/20 0.32
TSHR P16473 1/20 0.32
CACNA1G O43497 2/20 0.31
ADRB2 P07550 1/20 0.31
ADRB1 P08588 1/20 0.31
ADRB3 P13945 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA4 P43681 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9699602 0.88 MME (0.32) NAAAEDNRBEDNRA
SCHEMBL9698268 0.88 NAAA (0.31) NAAAEDNRBEDNRA
SCHEMBL10392875 0.86 VDR (0.31) NAAA
SCHEMBL9700881 0.85 S1PR2 (0.31) NAAA
SCHEMBL9699638 0.77 EBP (0.36)
SCHEMBL10394793 0.77 CYP3A4 (0.32) ALDH1A1CYP2D6CYP2C9CYP2C19
SCHEMBL10694561 0.72 SPHK2 (0.31) ALDH1A1HTT
Bromide SCHEMBL9718283 0.71 IDO1 (0.37)
SCHEMBL9813460 0.70 CYP4F2 (0.40) ALDH1A1TSHR
SCHEMBL9699643 0.68 MEN1 (0.30) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5106991-A Geminally substituted thiaheterocyclic carboxylic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1992-04-21 US disclosed
US-4975452-A Geminally substituted thiaheterocyclic carboxylic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1990-12-04 US disclosed