SCHEMBL9701351

SCHEMBL9701351

CNCC1Cn2c(C)cc3cccc(c32)O1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CASR P41180 11/20 0.37
HTR6 P50406 1/20 0.34
SLC6A4 P31645 5/20 0.34
CYP2D6 P10635 4/20 0.33
SLC6A2 P23975 4/20 0.33
SLC6A3 Q01959 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700002 0.83 HPGD (0.34) KDM4EALDH1A1HPGDHSD17B10CASR
SCHEMBL9701706 0.79 SLC6A4 (0.36) KDM4EALDH1A1HPGDHSD17B10SLC6A4
SCHEMBL9700179 0.79 ADRA2A (0.43)
SCHEMBL9699368 0.77 HRH3 (0.46)
SCHEMBL9700364 0.76 ADRA2A (0.35)
SCHEMBL9699053 0.70 CASR (0.35) CASRHTR6SLC6A4CYP2D6SLC6A2
SCHEMBL9699321 0.67 HTR6 (0.43) CASRHTR6
SCHEMBL9532833 0.65 CASR (0.59) CASRHTR6
SCHEMBL18258200 0.64 MCL1 (0.48)
Hydrochloric Acid SCHEMBL9455227 0.64 CASR (0.58) CASRHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed