SCHEMBL9701648

SCHEMBL9701648

COc1cccc2c1OCC(CN1CCCNCC1)N2N=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
HTR7 P34969 3/20 0.40
HTR1A P08908 5/20 0.39
ADRA1A P35348 5/20 0.39
ADRA1B P35368 3/20 0.39
ADRA1D P25100 2/20 0.39
HTR3A P46098 4/20 0.39
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
ADRB1 P08588 1/20 0.39
DRD2 P14416 1/20 0.39
CYP2C19 P33261 1/20 0.39
DRD3 P35462 1/20 0.39
HTR6 P50406 1/20 0.39
HTR3D Q70Z44 1/20 0.39
HTR3C Q8WXA8 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
ADRA2A P08913 1/20 0.37
ADRA2B P18089 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9699253 0.91 ADRA2A (0.42) HTR1AADRA1AADRA1BADRA1DDRD2
SCHEMBL9701674 0.91 ADRA2A (0.42) HTR1AADRA1AADRA1BADRA1DDRD2
SCHEMBL9700406 0.86 ADRB1 (0.38) LMNAMAPTHTR1AHTR3AADRB1
SCHEMBL9699287 0.85 HTR7 (0.40) LMNAMAPTHTR7HTR1AADRA1A
SCHEMBL9700405 0.85 ADRA2A (0.43) HTR1AADRA1AADRA1BADRA1DDRD2
SCHEMBL9699344 0.84 ADRA1A (0.42) HTR1AADRA1AADRA1BADRA1DDRD2
SCHEMBL9701645 0.78 HTR2C (0.35) LMNAMAPTHTR7HTR3AHTR3E
SCHEMBL9699276 0.78 ADRA2A (0.35) HTR7HTR1AADRA1AADRA1BADRA1D
SCHEMBL9701394 0.76 ADRA1A (0.36) ADRA1AADRA1BADRA1DDRD2ADRA2A
SCHEMBL9699297 0.75 NOTUM (0.38) ADRA1AADRA1BADRA1DDRD2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed