SCHEMBL9701645

SCHEMBL9701645

COc1cccc2c1OCC(CC1CNCCCN1)N2N=O

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.35
HTR2B P41595 5/20 0.35
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
ADRB1 P08588 1/20 0.32
DRD2 P14416 1/20 0.32
CYP2C19 P33261 1/20 0.32
DRD3 P35462 1/20 0.32
HTR3A P46098 1/20 0.32
HTR6 P50406 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
HTR2A P28223 3/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
HTR7 P34969 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700400 0.86 HTR2A (0.34) HTR2CHTR2BHTR6HTR2A
SCHEMBL9699281 0.85 HTR2C (0.37) HTR2CHTR2BCHRNB4CHRNA3HTR3E
SCHEMBL9701648 0.78 LMNA (0.41) HTR2CHTR2BHTR3EHTR3BADRB1
SCHEMBL9699276 0.77 ADRA2A (0.35) HTR2CHTR2BHTR2AHTR7
SCHEMBL9699253 0.75 ADRA2A (0.42) HTR2CDRD2DRD3HTR2A
SCHEMBL9701674 0.75 ADRA2A (0.42) HTR2CDRD2DRD3HTR2A
SCHEMBL9701394 0.75 ADRA1A (0.36) DRD2
SCHEMBL9701640 0.74 CHRNB4 (0.38) HTR2CHTR2BCHRNB4CHRNA3HTR2A
SCHEMBL9700405 0.72 ADRA2A (0.43) HTR2CDRD2DRD3HTR2A
SCHEMBL9699316 0.72 HTR2A (0.33) HTR2CHTR2BHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed