SCHEMBL9701976

SCHEMBL9701976

COC(=O)C(N)Cc1cc2nccnc2cc1CP(=O)(OC)OC

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.33
GRIN3B O60391 2/20 0.32
GRIN1 Q05586 2/20 0.32
GRIN2C Q14957 2/20 0.32
MAPT P10636 3/20 0.32
MEN1 O00255 2/20 0.32
POLB P06746 2/20 0.32
KMT2A Q03164 2/20 0.32
KDM4E B2RXH2 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
TP53 P04637 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ARHGEF12 Q9NZN5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700809 0.72
SCHEMBL9701943 0.70 KDM4E (0.38) KMT2AKDM4EL3MBTL1
SCHEMBL29039963 0.69 NLRP3 (0.41) ALDH1A1KMT2A
SCHEMBL6495560 0.69 LOXL2 (0.47) ALDH1A1MAPTKDM4E
Hydrochloric Acid SCHEMBL6495555 0.68 LOXL2 (0.46) ALDH1A1MAPTKDM4E
Hydrochloric Acid SCHEMBL6495563 0.68 LOXL2 (0.46) ALDH1A1MAPTKDM4E
SCHEMBL25919492 0.65 ALDH1A1 (0.39) ALDH1A1KMT2A
SCHEMBL28572795 0.65 PTGS2 (0.35) ALDH1A1GRIN3BGRIN1GRIN2CMEN1
SCHEMBL29671111 0.65 PTGS2 (0.35) ALDH1A1GRIN3BGRIN1GRIN2CMEN1
SCHEMBL7421530 0.65 SMN1; SMN2 (0.33) ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992014740-A1 QUINOXALINE PHOSPHONO-AMINO ACIDS AMERICAN HOME PRODUCTS CORPORATION (US) 1992-09-03 WO disclosed
US-5118675-A Therapy for central nervous system disorders AMERICAN HOME PRODUCTS CORPORATION (US) 1992-06-02 US disclosed