SCHEMBL9703378

SCHEMBL9703378

CCOC(=O)c1cn2c3c(c(Cl)c(F)cc3c1=O)C(=O)CC2CC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.45
STAT3 P40763 2/20 0.43
KMT2A Q03164 2/20 0.42
KDM4E B2RXH2 3/20 0.42
HPGD P15428 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HSD17B10 Q99714 2/20 0.42
CNR1 P21554 2/20 0.41
CNR2 P34972 2/20 0.41
HTT P42858 1/20 0.39
CYP2C19 P33261 1/20 0.39
POLB P06746 2/20 0.37
BAZ2B Q9UIF8 1/20 0.36
BAZ2A Q9UIF9 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
LMNA P02545 1/20 0.36
TOP2A P11388 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9703781 0.89 ADRB2 (0.46) ADRB2STAT3KMT2AKDM4EHPGD
SCHEMBL9704658 0.88 ALDH1A1 (0.44) KMT2AKDM4EHPGDALDH1A1HSD17B10
SCHEMBL9703919 0.83 MEN1 (0.48) ADRB2STAT3KMT2AKDM4EHPGD
SCHEMBL10646921 0.83 MAOB (0.34) ADRB2KDM4EALDH1A1HSD17B10CNR1
SCHEMBL9703608 0.83 KDM4E (0.42) ADRB2STAT3KMT2AKDM4EHPGD
SCHEMBL9704598 0.79 STAT3 (0.50) ADRB2STAT3KMT2AKDM4EHPGD
SCHEMBL9704619 0.79 BAZ2B (0.40) ADRB2STAT3KMT2AKDM4EHPGD
SCHEMBL5704396 0.78 ADRB2 (0.64) ADRB2STAT3KMT2AKDM4EHPGD
SCHEMBL9703892 0.78 TOP2A (0.40) ADRB2KMT2AKDM4EHPGDALDH1A1
SCHEMBL9703281 0.77 KDM4E (0.39) KDM4EHPGDALDH1A1HSD17B10CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0203795-B1 Benzo [i,j] quinolizine-2-carboxylic acid derivatives, the salts and their hydrates, pharmaceutical compositions thereof, and process for preparing the same TOKYO TANABE COMPANY LIMITED (JP) 1992-07-29 EP disclosed
US-4720495-A Benzo[ij]quinolizine-2-carboxylic acids useful for treating bacterial infection TOKYO TANABE CO. LIMITED (JP) 1988-01-19 US disclosed
EP-0203795-A2 Benzo [i,j] quinolizine-2-carboxylic acid derivatives, the salts and their hydrates, pharmaceutical compositions thereof, and process for preparing the same TOKYO TANABE COMPANY LIMITED (JP) 1986-12-03 EP disclosed