SCHEMBL9707422

SCHEMBL9707422

COC(C)n1c(=O)c2c(nc(C(C)C)n2Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n(CCc2ccccc2)c1=O

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.37
CRHBP P24387 2/20 0.37
CRHR2 Q13324 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
MCOLN3 Q8TDD5 1/20 0.37
AGTR1 P30556 4/20 0.37
AGTR2 P50052 2/20 0.37
LMNA P02545 2/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA1 P30542 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707769 0.92 ADORA3 (0.39) AGTR1AGTR2ADORA3ADORA1
SCHEMBL9708556 0.92 ADORA3 (0.42) MAPTCRHBPCRHR2NPSR1MCOLN3
SCHEMBL9708566 0.91 AGTR1 (0.38) MAPTCRHBPCRHR2NPSR1MCOLN3
SCHEMBL9707685 0.91 PPARG (0.35) AGTR1AGTR2
SCHEMBL9707862 0.91 PPARG (0.37)
SCHEMBL9707902 0.90 HPGD (0.43) MAPTCRHBPCRHR2NPSR1MCOLN3
SCHEMBL9707857 0.90 ALDH1A1 (0.38) MAPTALDH1A1SMN1; SMN2
SCHEMBL9708052 0.90 AGTR1 (0.40) AGTR1AGTR2
SCHEMBL9707419 0.90 ADORA3 (0.42) AGTR1LMNAALDH1A1TSHRSMN1; SMN2
SCHEMBL9708021 0.90 ADORA3 (0.42) AGTR1LMNAALDH1A1TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed