SCHEMBL9707857

SCHEMBL9707857

COC(C)n1c(=O)c2c(nc(C(C)C)n2Cc2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n(C)c1=O

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
USP1 O94782 3/20 0.37
DPP4 P27487 1/20 0.37
BRAF P15056 1/20 0.36
PIK3CG P48736 1/20 0.36
MAPT P10636 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708044 0.94 ALDH1A1 (0.38) ALDH1A1POLBUSP1MAPTSMN1; SMN2
SCHEMBL9707862 0.94 PPARG (0.37) USP1
SCHEMBL9707769 0.91 ADORA3 (0.39)
SCHEMBL9707685 0.91 PPARG (0.35)
SCHEMBL9708049 0.91 USP1 (0.34) USP1
SCHEMBL9707571 0.91 ALDH1A1 (0.38) ALDH1A1POLBDPP4BRAFPIK3CG
SCHEMBL9707422 0.90 MAPT (0.37) ALDH1A1MAPTSMN1; SMN2
SCHEMBL9707977 0.90 ALDH1A1 (0.44) ALDH1A1POLBDPP4MAPTSMN1; SMN2
SCHEMBL9708038 0.90 AGTR1 (0.35) USP1
SCHEMBL9708607 0.90 DPP4 (0.38) USP1DPP4BRAFPIK3CGMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed