SCHEMBL9707625

SCHEMBL9707625

Cc1nc2[nH]c(=O)n(CCc3ccccc3)c(=O)c2n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
HPGD P15428 1/20 0.41
AGTR1 P30556 6/20 0.39
AGTR2 P50052 4/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
RGS12 O14924 1/20 0.39
USP2 O75604 1/20 0.39
MAPT P10636 1/20 0.39
MCOLN3 Q8TDD5 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
ADORA2B P29275 1/20 0.38
PPARG P37231 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708605 0.92 ADORA2B (0.42) AGTR1AGTR2ADORA3ADORA2B
SCHEMBL9708298 0.90 ADORA2B (0.40) KDM4EHPGDAGTR1AGTR2MEN1
SCHEMBL9708519 0.90 DCTPP1 (0.42) KDM4EHPGDAGTR1AGTR2MEN1
SCHEMBL9707975 0.90 AGTR1 (0.42) AGTR1AGTR2ADORA2B
SCHEMBL9707747 0.89 KDM4E (0.44) KDM4EHPGDAGTR1AGTR2ADORA2B
SCHEMBL9707424 0.89 AGTR1 (0.44) AGTR1AGTR2
SCHEMBL9708226 0.89 AGTR1 (0.38) AGTR1AGTR2MAPTMCOLN3ADORA3
SCHEMBL9708252 0.88 ADORA3 (0.42) KDM4EHPGDAGTR1AGTR2ADORA3
SCHEMBL9707499 0.88 MEN1 (0.39) AGTR1AGTR2MEN1KMT2AADORA2B
SCHEMBL9707884 0.88 AGTR1 (0.49) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed