SCHEMBL9708519

SCHEMBL9708519

COCCn1c(=O)[nH]c2nc(C)n(Cc3ccc(-c4ccccc4-c4nnn[nH]4)cc3)c2c1=O

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DCTPP1 Q9H773 1/20 0.42
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 4/20 0.41
PKM P14618 1/20 0.41
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
PPARG P37231 3/20 0.38
GAA P10253 1/20 0.38
RECQL P46063 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
AGTR1 P30556 1/20 0.37
AGTR2 P50052 1/20 0.37
USP1 O94782 1/20 0.37
HPGD P15428 3/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708605 0.91 ADORA2B (0.42) AGTR1AGTR2
SCHEMBL9707572 0.90 AGTR1 (0.41) DCTPP1KDM4EALDH1A1PKMPPARG
SCHEMBL9707625 0.90 KDM4E (0.41) KDM4EMEN1KMT2APPARGAGTR1
SCHEMBL9708640 0.90 USP1 (0.42) DCTPP1KDM4EALDH1A1PKMMEN1
SCHEMBL9708298 0.89 ADORA2B (0.40) KDM4EMEN1KMT2AAGTR1AGTR2
SCHEMBL9708254 0.89 AGTR1 (0.43) PPARGAGTR1AGTR2
SCHEMBL9707673 0.88 KDM4E (0.37) DCTPP1KDM4EALDH1A1PKMMEN1
SCHEMBL9707747 0.88 KDM4E (0.44) DCTPP1KDM4EAGTR1AGTR2HPGD
SCHEMBL9708271 0.88 AGTR1 (0.42) KMT2APPARGSMN1; SMN2AGTR1AGTR2
SCHEMBL9707446 0.87 AGTR1 (0.47) PPARGAGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed