SCHEMBL9707658

SCHEMBL9707658

CC(C)(C)Cc1nc2c(c(=O)[nH]c(=O)n2CC2CC2)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.41
MEN1 O00255 5/20 0.41
TPH1 P17752 10/20 0.39
TPH2 Q8IWU9 10/20 0.39
AGTR1 P30556 1/20 0.39
AGTR2 P50052 1/20 0.39
ALDH1A1 P00352 2/20 0.38
HTT P42858 2/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
NPSR1 Q6W5P4 2/20 0.38
TSHR P16473 1/20 0.37
CNR2 P34972 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708230 0.91 KMT2A (0.45) KMT2AMEN1TPH1TPH2AGTR1
SCHEMBL9708379 0.90 MEN1 (0.46) KMT2AMEN1TPH1TPH2AGTR1
SCHEMBL9707269 0.90 MEN1 (0.51) KMT2AMEN1TPH1TPH2
SCHEMBL9707770 0.89 AGTR1 (0.50) KMT2AMEN1AGTR1AGTR2
SCHEMBL9707595 0.88 PDE5A (0.47) AGTR1AGTR2
SCHEMBL9707703 0.88 TPH1 (0.49) KMT2AMEN1TPH1TPH2ALDH1A1
SCHEMBL9708645 0.88 ALDH1A1 (0.42) KMT2AMEN1AGTR1AGTR2ALDH1A1
SCHEMBL9707461 0.88 AGTR1 (0.48) KMT2AMEN1AGTR1AGTR2
SCHEMBL9707751 0.88 ADORA3 (0.40) AGTR1AGTR2CNR2
SCHEMBL9708617 0.88 MEN1 (0.42) KMT2AMEN1TPH1TPH2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed