SCHEMBL9708044

SCHEMBL9708044

COC(C)n1c(=O)n(C)c(=O)c2c1nc(C(C)C)n2Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
POLB P06746 1/20 0.38
USP1 O94782 3/20 0.38
MAPT P10636 2/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
HIF1A Q16665 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707857 0.94 ALDH1A1 (0.38) ALDH1A1POLBUSP1MAPTSMN1; SMN2
SCHEMBL9707862 0.93 PPARG (0.37) USP1
SCHEMBL9707505 0.91 ADORA3 (0.40)
SCHEMBL9707740 0.91 PPARG (0.35)
SCHEMBL9708111 0.91 ALDH1A1 (0.39) ALDH1A1POLBMAPTHPGDSMN1; SMN2
SCHEMBL9707977 0.91 ALDH1A1 (0.44) ALDH1A1POLBMAPTSMN1; SMN2HIF1A
SCHEMBL9707896 0.90 DPP4 (0.37) ALDH1A1USP1MAPTHPGDSMN1; SMN2
SCHEMBL9708894 0.90 AGTR1 (0.35) USP1
SCHEMBL9707440 0.89 AGTR1 (0.41) ALDH1A1POLBSMN1; SMN2ALOX15HSD17B10
SCHEMBL9708014 0.89 AGTR1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed