SCHEMBL9707977

SCHEMBL9707977

CC(C)c1nc2c(c(=O)n(C)c(=O)n2C)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
HIF1A Q16665 1/20 0.44
ALOX15 P16050 1/20 0.44
HSD17B10 Q99714 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 4/20 0.43
TSHR P16473 4/20 0.43
NPSR1 Q6W5P4 3/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 2/20 0.43
POLB P06746 1/20 0.43
PCSK9 Q8NBP7 1/20 0.43
DPP4 P27487 1/20 0.43
USP2 O75604 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ATM Q13315 1/20 0.42
THRB P10828 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9708010 0.92 MAPT (0.41) MAPTPOLBDPP4MEN1KMT2A
SCHEMBL9708826 0.92 HPGD (0.41) ATM
SCHEMBL9707347 0.91 RAB9A (0.44) SMN1; SMN2HSD17B10LMNAMAPTTSHR
SCHEMBL9708648 0.91 ADORA1 (0.42) MAPTDPP4
SCHEMBL9708391 0.91 PDE1A (0.44) SMN1; SMN2LMNATSHRNPSR1
SCHEMBL9707814 0.91 ADORA3 (0.42) SMN1; SMN2LMNA
SCHEMBL9708044 0.91 ALDH1A1 (0.38) ALDH1A1SMN1; SMN2HIF1AALOX15HSD17B10
SCHEMBL9707660 0.91 USP1 (0.39) ALDH1A1SMN1; SMN2ALOX15HSD17B10LMNA
SCHEMBL9708188 0.91 USP1 (0.39) ALDH1A1SMN1; SMN2ALOX15HSD17B10LMNA
SCHEMBL9707902 0.90 HPGD (0.43) ALDH1A1SMN1; SMN2ALOX15HSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed