SCHEMBL9708310

SCHEMBL9708310

CC(C)Cn1c(=O)c2c(nc(C(C)C)n2Cc2ccc(-c3ccccc3)c(-c3nnn[nH]3)c2)n(C)c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ADORA1 P30542 5/20 0.40
ADORA3 P0DMS8 4/20 0.40
ADORA2A P29274 3/20 0.40
ADORA2B P29275 3/20 0.40
LMNA P02545 3/20 0.39
NPSR1 Q6W5P4 2/20 0.39
MAPK1 P28482 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
CASP1 P29466 2/20 0.39
TSHR P16473 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HIF1A Q16665 1/20 0.38
HTT P42858 1/20 0.38
CASP7 P55210 1/20 0.38
HSD17B10 Q99714 1/20 0.38
BRAF P15056 1/20 0.37
PIK3CG P48736 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707347 0.91 RAB9A (0.44) RAB9AMEN1KMT2AADORA1ADORA3
SCHEMBL9708591 0.91 ADORA1 (0.40) ADORA1ADORA3ADORA2AADORA2BMAPK1
SCHEMBL9708262 0.87 HPGD (0.42) MEN1KMT2ALMNANPSR1MAPK1
SCHEMBL9708010 0.85 MAPT (0.41) RAB9AMEN1KMT2AADORA1ADORA3
SCHEMBL9707680 0.85 ADORA3 (0.43) MEN1KMT2AADORA1ADORA3ADORA2A
SCHEMBL9708391 0.85 PDE1A (0.44) LMNANPSR1SMN1; SMN2CASP1TSHR
SCHEMBL9708251 0.84 ALDH1A1 (0.37) MEN1KMT2ALMNANPSR1SMN1; SMN2
SCHEMBL9708819 0.84 ADORA3 (0.44) ADORA1ADORA3ADORA2AADORA2B
SCHEMBL9708697 0.84 ADORA3 (0.39) MEN1KMT2AADORA1ADORA3ADORA2A
SCHEMBL9708654 0.83 ADORA3 (0.42) ADORA1ADORA3ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed